Cathepsin X-IN-1

CAS No. 2418577-51-0

Cathepsin X-IN-1( —— )

Catalog No. M35476 CAS No. 2418577-51-0

Cathepsin X-IN-1 (compound 25) is a potent Cathepsin X inhibitor (IC50 = 7.13 μM) that reduces PC-3 cell migration with low cytotoxicity .

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 55 Get Quote
10MG 93 Get Quote
25MG 181 Get Quote
50MG 297 Get Quote
100MG 419 Get Quote
200MG 583 Get Quote
500MG Get Quote Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    Cathepsin X-IN-1
  • Note
    Research use only, not for human use.
  • Brief Description
    Cathepsin X-IN-1 (compound 25) is a potent Cathepsin X inhibitor (IC50 = 7.13 μM) that reduces PC-3 cell migration with low cytotoxicity .
  • Description
    Cathepsin X-IN-1 (compound 25) is a potent Cathepsin X inhibitor with an IC50 of 7.13 μM. Cathepsin X-IN-1 decreases PC-3 cell migration with low cytotoxic.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Proteasome/Ubiquitin
  • Target
    Cysteine Protease
  • Recptor
    Cysteine Protease
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    2418577-51-0
  • Formula Weight
    315.35
  • Molecular Formula
    C15H13N3O3S
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?DMSO : ≥ 100 mg/mL (317.11 mM; )H2O : ≥ 4.85 mg/mL (15.38 mM)
  • SMILES
    O=C(CSc1nccn1CC#N)c1ccc2OCCOc2c1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Fonovi? UP, et al. Structure-activity relationships of triazole-benzodioxine inhibitors of cathepsin X. Eur J Med Chem. 2020 May 1;193:112218.?
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